These are medication that serve as a "partial agonists" for the
treatment of opiate and narcotic abuse. Suboxone is a new medication FDA approved for the treatment of opiate dependence. It has no
desirable euphoria or "high", even if taken in larger doses,
because it does not fully activate the body's opiate receptors. Think
of it as having a
"ceiling effect" or a "governor" or built-in limiter. This makes buprenorphine very
safe because it is difficult to "overdose". Buprenorphine also
interferes with the ability of other opiates to make someone euphoric or "high" because
it is "sticky" and other opiates have to displace it off the receptors before
they can work.
The Drug Enforcement Agency (DEA) requires special training
and special "waiver" in order to prescribe
Suboxone. There is also a federally designated limit to the number of
patients a practitioner can treat, making access to Suboxone a precious
limited resource.
(Suboxone is buprenorphine mixed with another drug that is an INACTIVE
INGREDIENT when taken as prescribed. This drug, Naloxone, is an
antagonist or "antidote" to opiates. When taken sublingual or orally
it is essentially not absorbed into the blood, When Suboxone is taken
sublingually as directed, this other ingredient has no significant effect. However, if Suboxone is crushed and "cooked" and injected intravenously,
the Naloxone RIPS EVERY OPIATE OFF EVERY OPIATE RECEPTOR in the body!
This would cause immediate severe withdrawal and be extremely unpleasant!
This other drug is mixed in ONLY to ruin Suboxone abuse for needle users.
Active opiate addicts will avoid injecting Suboxone as if it were a poison!)